Big Lecture Hall, Department of Chemistry
University of Basel, St. Johanns-Ring 19
May 22, 2014, 13.30-17.45
This year's annual mini-symposium organized by the Division of Medicinal Chemistry & Chemical Biology of the Swiss Chemical Society is dedicated to the topic of Kinetics and Thermodynamics in Drug Discovery.
This free event is gathering five globally renowed experts in the field that will showcase the importance of this topic in drug discovery.
Program
| 13:30–13:35 | Introduction |
| 13:35–14:20 |
Gerhard Klebe, University of Marburg Correlation of Structure, Thermodynamics and Molecular Dynamics to Better Understand Drug Binding |
| 14:20–15:05 |
David Swinney, iRND3 Application of binding kinetics to drug discovery |
| 15:05–15:30 | Coffee Break |
| 15:30–16:15 |
Göran Dahl, AstraZeneca Pharmacokinetics and the drug-target residence time concept |
| 16:15–17:00 |
David Sykes, Novartis Institutes for Biomedical Research Exploring the relationship betweenb2 adrenoceptor drug binding affinity/kinetic constants and physicochemical parameters |
| 17:00–17:45 |
Russel Petter, Celgene Design and Optimization of Targeted Covalent Inhibitors |
Contact
Herr Dr. Nikolaus Stiefl
Novartis Pharma AG
Forum1, Novartis Campus
4056 Basel
David Spichiger, SCS
03.02.2014